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Dr fahad anti arrythmic drugs
1.
Antiarrhythmic Drugs-Overview
Dr. Fahad Azam Shifa College of Medicine
2.
Classification of antiarrhythmic
drugs Classification of drugs Mechanism of action IA Na+ channel blocker Qunidine, Procainamide IB Na+ channel blocker Lidocaine, Mexiletine IC Na+ channel blocker Flecainide, Propafenone II Beta receptor blocker Propanalol, Metoprolol III K+ channel blocker Amiodarone, Sotalol, IV Ca+ channel blocker Verapamil, Diltiazem, Nifedipine
3.
Conduction Pathways and
Velocity of Conduction • Conduction Pathway: SA node atrial muscle AV node Purkinjee fibers Ven. Muscle delay • Velocity: – Fast conducting fiber: • Purkinjee cell, Ventricular muscle, Atrial muscle – Slow conducting fiber: • AV node, SA node
4.
Classification
Mechanism of action of drugs IA Na+ channel blocker Qunidine, Procainamide IB Na+ channel blocker Lidocaine, Mexiletine IC Na+ channel blocker Flecainide, Propafenone II Beta receptor blocker Propanalol, Metoprolol III K+ channel blocker Amiodarone, Sotalol, IV Ca+ channel blocker Verapamil, Diltiazem, Nifedipine
5.
Intracellular
Extracellular Na Leak Na Pump K Pump K Diffusion
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